中文介紹：

THPTA（三羥丙基三唑基甲胺）是一種水溶性、非常有效的加速配體緊密協作，用于銅催化的炔烴-疊氮化物點擊化學(xué)反應(yīng)（CuAAC）有力扭轉。除了大大提高CuAAC的速率外資源配置，THPTA還最大限度地減少了對所探測細(xì)胞或生物體生理狀態(tài)的擾動大幅拓展，并通過進(jìn)一步降低催化劑配方中的Cu負(fù)載量實際需求，允許有效的生物偶聯(lián)與抑制細(xì)胞細(xì)胞毒性非常完善。水溶性THPTA配體允許整個反應(yīng)在水中運(yùn)行深入各系統，進(jìn)一步簡化了點擊化學(xué)創造性。

英文介紹：

THPTA (tris-hydroxypropyltriazolylmethylamine) is a water-soluble, very effective accelerating ligand for copper-catalyzed Alkyne-Azide click chemistry reactions (CuAAC). In addition to greatly enhancing the rate of CuAAC, THPTA minimizes perturbations to the physiological state of the cells or organisms probed and allows for the effective bioconjugation with suppressed cell cytotoxicity by further lowering Cu loading in the catalyst formulation. The water-soluble THPTA ligand further simplifies click chemistry by allowing the entire reaction to be run in water.

產(chǎn)品參數(shù)：

參考文獻(xiàn)：

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